找到约 5 条 “Valproic acid” 相关结果 (用时 0.127 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M1876 | Valproic acid sodium salt | 丙戊酸钠盐;敌白痉;德巴金 | HDAC |
Sodium valproate | |||
Valproic acid sodium salt (Sodium valproate)是一种HDAC抑制剂,IC50为0.4 mM,也抑制GABA-转氨酶或琥珀酸半醛脱氢酶。 | |||
M9054 | Valproic acid | 丙戊酸 | HDAC |
Erganyl; Stavzor; VPA | |||
Valproic acid (VPA) 是一种 HDAC 抑制剂,其IC50值的范围为0.5~2 mM。此外,Valproic acid 还能显著促进重编程。Valproic acid (VPA) 可以激活 Notch-1 信号。 | |||
M8204 | VAHA | VAHA | Others |
Hydroxamic acid derivatives of valproic acid exhibit anticonvulsant activity with no teratogenic activity in mouse neural tube defect model. | |||
M8845 | Valpromide | 丙戊酰胺 | Epoxide Hydrolase |
Valpromide (VPD) is a derivative of valproic acid (VPA) and is used as an antiepileptic drug. | |||
M8847 | Valnoctamide | 戊诺酰胺 | Others |
Valproic acid (VPA) and derivatives such as valpromide and valnoctamide are anti-convulsant, mood stabilizing drugs, believed to function as indirect GABA agonists by inhibiting the transamination of GABA. |
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